Catalytic highly enantioselective vinylogous Povarov reaction
نویسندگان
چکیده
منابع مشابه
Catalytic highly enantioselective vinylogous Povarov reaction.
The first example of a catalytic asymmetric vinylogous Povarov reaction is presented. 1-N-Acylamino-1,3-butadienes react selectively at their terminal double bond in the presence of a chiral phosphoric acid catalyst, delivering highly enantioenriched 1,2,3,4-tetrahydroquinolines bearing a synthetically versatile enecarbamate group at the 4-position.
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ژورنال
عنوان ژورنال: Chem. Commun.
سال: 2013
ISSN: 1359-7345,1364-548X
DOI: 10.1039/c2cc38002a